7 Bis(het)aryl-1,2,3-triazole quinuclidines as α7 nicotinic acetylcholine receptor ligands: Synthesis, structure affinity relationships, agonism activity, [F]-radiolabeling and PET study in rats.

8 Discovery of 1,2,3-triazole-based fibroblast growth factor receptor modulators.

9 Emission Properties of Diblock Copolymers Composed of Poly(ethylene glycol) and Dense 1,2,3-Triazole Blocks.

10 Nickel-Catalyzed Coupling of N-Sulfonyl-1,2,3-triazole with H-Phosphine Oxides: Stereoselective and Site-Selective Synthesis of α-Aminovinylphosphoryl Derivatives.

11 Design, Synthesis, and Structure-Activity Relationships of 1,2,3-Triazole Benzenesulfonamides as New Selective Leucine-Zipper and Sterile-α Motif Kinase (ZAK) Inhibitors.

12 Synthesis of a new series of 3-functionalised-1-phenyl-1,2,3-triazole sulfamoylbenzamides as carbonic anhydrase I, II, IV and IX inhibitors.

13 Facile Synthesis, Characterization of New Quinazolinones with Different Azo Compounds, 1,2,3-Triazole Moieties and Evaluation Their Anti-bacterial Activity.

14 Synthesis and biological evaluation of benzimidazole-linked 1,2,3-triazole congeners as agents.

15 Acid-mediated synthesis of fully substituted 1,2,3-triazoles: Multicomponent coupling reactions, mechanistic study, synthesis of serine hydrolase inhibitor and its derivatives

16 Metal-free C-N- and N-N-bond formation: Synthesis of 1,2,3-triazoles from ketones, N-tosylhydrazines, and amines in one pot

17 Enamine/enolate-mediated organocatalytic azide- Carbonyl [3+2] cycloaddition reactions for the synthesis of densely functionalized 1,2,3-triazoles

18 Regioselective click chemistry for construction of arylpiperazinyl 1,2,3-triazole derivative libraries as dopamine D<inf>4</inf>/D<inf>3</inf> receptor ligands

19 Synthesis of N -acylamidines via rhodium-catalyzed reaction of nitrosobenzene derivatives with N -sulfonyl-1,2,3-triazoles

20 'Green' synthesis of 1,4-disubstituted 5-iodo-1,2,3-triazoles under neat conditions, and an efficient approach of construction of 1,4,5-trisubstituted 1,2,3-triazoles in one pot

21 An enolate-mediated organocatalytic Azide-Ketone [3+2]-cycloaddition reaction: Regioselective high-yielding synthesis of fully decorated 1,2,3-Triazoles

22 An efficient protocol for domino one pot synthesis of 1,2,3-triazoles from natural organic acids and phenols

23 Copper nanoparticles supported on agarose as a bioorganic and degradable polymer for multicomponent click synthesis of 1,2,3-triazoles under low copper loading in water

24 Regioselective one-pot synthesis of 1,4-disubstituted 1,2,3-triazole derivatives

25 Enhanced sensory response of quaterthiophene bearing 1,2,3-triazole moiety to explosives

26 Diastereoselective synthesis of tetrahydrofurano- and tetrahydropyrano-dihydropyrroles containing N,O-acetal moieties via rhodium-catalyzed transannulation of N-sulfonyl-1,2,3-triazoles with oxacycloalkenes

27 1H-1,2,3-triazole tethered isatin-ferrocene conjugates: Synthesis and in vitro antimalarial evaluation

28 Design and synthesis of pironetin analogue/combretastatin A-4 hybrids containing a 1,2,3-triazole ring and evaluation of their cytotoxic activity

29 Rhodium(II)-catalyzed stereocontrolled synthesis of 2-tetrasubstituted saturated heterocycles from 1-sulfonyl-1,2,3-triazoles

30 Facile synthesis of pyrroles via Rh(II)-catalyzed transannulation of 1-tosyl-1,2,3-triazoles with silyl or alkyl enol ethers

31 Polystyrene resin-supported CuI-cryptand 22 complex: A highly efficient and reusable catalyst for three-component synthesis of 1,4-disubstituted 1,2,3-triazoles under aerobic conditions in water

32 Discovery and biological evaluation of novel 6,7-disubstituted-4-(2-fluorophenoxy)quinoline derivatives possessing 1,2,3-triazole-4-carboxamide moiety as c-Met kinase inhibitors

33 Extraction Properties of 1,2,3-Triazole Modified Carbamoylmethylphosphine Oxide in Nitric Acid Media

34 P -toluenesulfonic acid mediated 1,3-dipolar cycloaddition of nitroolefins with NaN <inf>3</inf> for synthesis of 4-Aryl- NH -1,2,3-triazoles

35 Rhodium(III)-Catalyzed Direct C-H Alkylation of 2-Aryl-1,2,3-triazole N-Oxides with Maleimides

36 N-Heterocyclic carbene–copper complex supported on ionic liquid-modified graphene oxide: versatile catalyst for synthesis of (i) 1,2,3-triazole and (ii) propargylamine derivatives

37 Room-temperature oxidative Suzuki coupling reaction of 1,2,3-triazole N-oxides

38 Iridium(III)-Catalyzed Direct C-H Sulfonamidation of 2-Aryl-1,2,3-triazole N-Oxides with Sulfonyl Azides

39 Palladium-catalyzed highly regioselective oxidative homocoupling of 1,2,3-triazole N-oxides

40 NiSO<inf>4</inf>-catalyzed C-H activation/C-S cross-coupling of 1,2,3-triazole N-oxides with thiols

41 Highly regioselective arylation of 1,2,3-triazole N-oxides with sodium arenesulfinates via palladium-catalyzed desulfitative cross-coupling reaction

42 Copper-catalyzed direct amination of 1,2,3-triazole N-oxides by C-H activation and C-N coupling

43 Site-selective direct arylation of 1,2,3-triazole N-oxides

44 Palladium-catalyzed olefination and arylation of 2-substituted 1,2,3-triazole N -oxides

45 <sup>14</sup> N and <sup>15</sup> N NMR spectroscopy of 2-methyl-4,5-dinitro-1,2,3-triazole and of substituted 2-methyl-4(5)-nitro-1,2,3-triazole 1-oxides

46 Intramolecular cyclization of 1,2-bis(N-alkoxy-N-nitrosoamino)alkanes: A unique route to 4,5-dihydro-1,2,3-triazole 2-oxides

47 Unexpected transformation of 1,2-bis(N-methoxy-N-nitrosoamino)cycloalkanes: First synthesis of 4,5-dihydro-1,2,3-triazole 2-oxides

48 1,2,3-Triazole N-Oxides. II. Synthesis of Substituted 4(5)-Ethoxycarbonyl-1,2,3-triazole N-Oxides

49 Preparation of 1-hydroxypyrazoles and 1-hydroxy-1,2,3-triazoles by dealkylation of pyrazole and triazole N-oxides

50 Extended tandem reactions of 2H-1,2,3-triazole N-oxides with dialkyl acetylenedicarboxylates and N-phenylmaleimide: Substituted monocyclic 2,5-dihydro-1,2,3-triazines and new tetrahydrofuro[2,3-d]-1,2,3-triazoles. Azolium 1,3-dipoles. Part 5.

51 2,5-Dihydro-1,2,3-triazine derivatives from attempted 1,3-dipolar cycloaddition of 1,2,3-triazole N-oxides with dimethyl acetylenedicarboxylate: A new ring expansion

52 Synthesis of new thiazolyl-pyrazolyl-1,2,3-triazole derivatives as potential antimicrobial agents.

53 Synthesis of novel (R)-4-fluorophenyl-1H-1,2,3-triazoles: A new class of α-glucosidase inhibitors.

54 Identification of potent triazolylpyridine nicotinamide phosphoribosyltransferase (NAMPT) inhibitors bearing a 1,2,3-triazole tail group.

55 Crystal structure of 1-anilino-5-methyl-1-1,2,3-triazole-4-carb-oxy-lic acid monohydrate.

56 Efficient synthesis, spectroscopic characterization and DFT based studies of novel 1-amide 4-sulfonamide-1,2,3-triazole derivatives

57 Design and microwave-assisted synthesis of dimers of 1,5-benzodiazepine-1,2,3-triazole hybrids bearing alkyl/aryl spacers and their biological assessment

58 Design, synthesis and antibacterial evaluation of novel 15-membered 11a-azahomoclarithromycin derivatives with the 1, 2, 3-triazole side chain

59 Cu(OTf)<inf>2</inf>-Catalyzed 1,2,3-triazole-ring-controlled selective phenolic O–H bond methylthiomethylation

60 Synthesis and biological evaluation of bergenin-1,2,3-triazole hybrids as novel class of anti-mitotic agents

61 NiSO4-catalyzed C-H activation/C-S cross-coupling of 1,2,3-triazole N-oxides with thiols.

62 Electrophilic and nucleophilic substitution in the triazole N-oxides and N-methoxytriazolium salts: Preparation of substituted 1,2,3-triazoles

63 Photochemistry of azole n-oxides. III photoinduced ring expansion of 2h-1, 2, 3-triazole n-oxides

64 Conversion of α-azoxyoximes to 2H-1,2,3-triazole N-oxide derivatives

65 The infrared spectra of 1,2,3-triazole N-oxides

66 Biscoumarin-1,2,3-triazole hybrids as novel anti-diabetic agents: Design, synthesis, in vitro α-glucosidase inhibition, kinetic, and docking studies.

67 A General Proline Catalyzed Synthesis of 4,5-Disubstituted N-Sulfonyl-1,2,3-Triazoles from 1,3-Dicarbonyl Compounds and Sulfonyl Azide.

68 Gatifloxacin-1,2,3-triazole-isatin hybrids and their antimycobacterial activities.

69 New amide linked dimeric 1,2,3-triazoles bearing aryloxy scaffolds as a potent antiproliferative agents and EGFR tyrosine kinase phosphorylation inhibitors.

70 Complexes of (η(6)-benzene)ruthenium(II) with 1,4-bis(phenylthio/seleno-methyl)-1,2,3-triazoles: synthesis, structure and applications in catalytic activation of oxidation and transfer hydrogenation.

71 Design, Synthesis and Anti-Platelet Aggregation Activity Study of Ginkgolide-1,2,3-triazole Derivatives

72 Semi-synthesis of β-keto-1,2,3-triazole derivatives from ethinylestradiol and evaluation of the cytotoxic activity.

73 Copper-Catalyzed Three-Component Reaction of Alkynes, TMSN, and Ethers: Regiocontrollable Synthesis of N- and N-Oxyalkylated 1,2,3-Triazoles.

74 Nucleoside dimers analogues with a 1,2,3-triazole linkage: conjugation of floxuridine and thymidine provides novel tools for cancer treatment. Part II

75 A click chemistry approach for the synthesis of cyclic ureido tethered coumarinyl and 1-aza coumarinyl 1,2,3-triazoles as inhibitors of Mycobacterium tuberculosis H37Rv and their in silico studies

76 Design, synthesis and antibacterial activity evaluation of moxifloxacin-amide-1,2,3-triazole-isatin hybrids

77 Catalyst-free facile synthesis of polycyclic indole/pyrrole substituted-1,2,3-triazoles

78 Ciprofloxacin-1,2,3-triazole-isatin hybrids tethered via amide: Design, synthesis, and in vitro anti-mycobacterial activity evaluation

79 New thiosemicarbazide-1,2,3-triazole hybrids as potent α-glucosidase inhibitors: Design, synthesis, and biological evaluation

80 Microwave-assisted synthesis of new pyrazole derivatives bearing 1,2,3-triazole scaffold as potential antimicrobial agents

81 1,2,3-Triazole-containing hybrids as potential anticancer agents: Current developments, action mechanisms and structure-activity relationships.

82 Synthesis of novel N-heterocyclic compounds containing 1,2,3-triazole ring system via domino, “click” and RDA reactions

83 Recent Advances in Transition-Metal-Catalyzed Denitrogenative Transformations of 1,2,3-Triazoles and Related Compounds

84 Fragmentation de Triazoles Sous L'Impact Electronique—II 1,2,3-Triazole

85 Synthesis of 4-aminoquinoline-1,2,3-triazole and 4-aminoquinoline-1,2,3-triazole-1,3,5-triazine Hybrids as Potential Antimalarial Agents

86 1,4-Diphenyl-5-Amino-1,2,3-Triazole and 4-Phenyl-5-Anilino-1,2,3-Triazole

87 Mesoionic 1,2,3-Triazoles and 1,2,3-Triazole Carbenes

88 “Click-Triazole” Coordination Chemistry: Exploiting 1,4-Disubstituted-1,2,3-Triazoles as Ligands

89 Synthesis of 1,4,5-Trisubstituted-1,2,3-triazoles by Copper-Catalyzed Cycloaddition-Coupling of Azides and Terminal Alkynes.

90 Synthesis of 1,4,5-trisubstituted-1,2,3-triazoles by copper-catalyzed cycloaddition-coupling of azides and terminal alkynes

91 ChemInform Abstract: Direct Access to 1,4-Disubstituted 1,2,3-Triazoles Through Organocatalytic 1,3-Dipolar Cycloaddition Reaction of α,β-Unsaturated Esters with Azides.

92 Direct access to 1,4-disubstituted 1,2,3-triazoles through organocatalytic 1,3-dipolar cycloaddition reaction of α,β-unsaturated esters with azides

93 ChemInform Abstract: Ln[N(SiMe3)2]3-Catalyzed Cycloaddition of Terminal Alkynes to Azides Leading to 1,5-Disubstituted 1,2,3-Triazoles: New Mechanistic Features.

94 Ln[N(SiMe3)2]3-catalyzed cycloaddition of terminal alkynes to azides leading to 1,5-disubstituted 1,2,3-triazoles: new mechanistic features

95 Potassium tert-Butoxide Promoted Cycloaddition Reaction for the Synthesis of 1,5-Disubstituted 1,2,3-Triazoles from Aromatic Azides and Trimethylsilyl-Protected Alkynes

96 ChemInform Abstract: Potassium tert-Butoxide Promoted Cycloaddition Reaction for the Synthesis of 1,5-Disubstituted 1,2,3-Triazoles from Aromatic Azides and Trimethylsilyl-Protected Alkynes.

97 A Microwave-Assisted Click Chemistry Synthesis of 1,4-Disubstituted 1,2,3-Triazoles via a Copper(I)-Catalyzed Three-Component Reaction.

98 Design, synthesis, in silico and in vitro antimicrobial screenings of novel 1,2,4-triazoles carrying 1,2,3-triazole scaffold with lipophilic side chain tether.

99 Selective C(sp)-H Halogenation of "Click" 4-Aryl-1,2,3-triazoles.

100 Synthesis, anti-inflammatory, bactericidal activities and docking studies of novel 1,2,3-triazoles derived from ibuprofen using click chemistry.

101 Synthesis of bi- and bis-1,2,3-triazoles by copper-catalyzed Huisgen cycloaddition: A family of valuable products by click chemistry.

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