| 31 |
Design, synthesis and biological evaluation of flexible and rigid analogs of 4H-1,2,4-triazoles bearing 3,4,5-trimethoxyphenyl moiety as new antiproliferative agents.
Ansari, Mahsa, Shokrzadeh, Mohammad, Karima, Saeed, Rajaei, Shima, Hashemi, Seyedeh Mahdieh, Mirzaei, Hassan, Fallah, Marjan, Emami, Saeed,
Vol. 93 pp. 103300
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2019 |
696
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| 7 |
Design, synthesis and anticervical cancer activity of new benzofuran-pyrazol-hydrazono- thiazolidin-4-one hybrids as potential EGFR inhibitors and apoptosis inducing agents.
Abbas, Hebat-Allah S, Abd El-Karim, Somaia S,
Vol. 89 pp. 103035
|
2019 |
695
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| 128 |
Design, synthesis and molecular docking of new pyrazole-thiazolidinones as potent anti-inflammatory and analgesic agents with TNF-α inhibitory activity.
Abd El-Karim, Somaia S, Mohamed, Hanaa S, Abdelhameed, Mohamed F, El-Galil E Amr, Abd, Almehizia, Abdulrahman A, Nossier, Eman S,
Vol. 111 pp. 104827
|
2021 |
678
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| 89 |
Design, synthesis, mechanistic studies and in silico ADME predictions of benzimidazole derivatives as novel antifungal agents.
Morcoss, Martha M, Abdelhafez, El Shimaa M N, Ibrahem, Reham A, Abdel-Rahman, Hamdy M, Abdel-Aziz, Mohamed, Abou El-Ella, Dalal A,
Vol. 101 pp. 103956
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2020 |
594
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| 8 |
Design, synthesis, modeling studies and biological screening of novel pyrazole derivatives as potential analgesic and anti-inflammatory agents.
Taher, Azza T, Mostafa Sarg, Marwa T, El-Sayed Ali, Nermeen R, Hilmy Elnagdi, Noha,
Vol. 89 pp. 103023
|
2019 |
573
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| 75 |
Design, synthesis and ADMET prediction of bis-benzimidazole as anticancer agent.
Rashid, Mohammad,
Vol. 96 pp. 103576
|
2020 |
568
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| 50 |
Design, synthesis, in vitro evaluation, molecular docking and ADME properties studies of hybrid bis-coumarin with thiadiazole as a new inhibitor of Urease.
Alomari, Munther, Taha, Muhammad, Imran, Syahrul, Jamil, Waqas, Selvaraj, Manikandan, Uddin, Nizam, Rahim, Fazal,
Vol. 92 pp. 103235
|
2019 |
519
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| 28 |
Design, synthesis and antibacterial activity evaluation of moxifloxacin-amide-1,2,3-triazole-isatin hybrids
Gao, F.
Vol. 91 pp. 103162
|
2019 |
511
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| 33 |
Design, synthesis and molecular docking of new N-4-piperazinyl ciprofloxacin-triazole hybrids with potential antimicrobial activity.
Mohammed, Hamada H H, Abdelhafez, El-Shimaa M N, Abbas, Samar H, Moustafa, Gamal A I, Hauk, Glenn, Berger, James M, Mitarai, Satoshi, Arai, Masayoshi, Abd El-Baky, Rehab M, Abuo-Rahma, Gamal El-Din A,
Vol. 88 pp. 102952
|
2019 |
509
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| 23 |
Design, synthesis, and molecular docking study of new piperazine derivative as potential antimicrobial agents.
Patil, Mahadev, Noonikara Poyil, Anurag, Joshi, Shrinivas D, Patil, Shivaputra A, Patil, Siddappa A, Bugarin, Alejandro,
Vol. 92 pp. 103217
|
2019 |
471
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| 63 |
Design and synthesis of novel Imidazo[2,1-b]thiazole derivatives as potent antiviral and antimycobacterial agents.
Gürsoy, Elif, Dincel, Efe Doğukan, Naesens, Lieve, Ulusoy Güzeldemirci, Nuray,
Vol. 95 pp. 103496
|
2019 |
455
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| 35 |
1,2,4-Triazole-based benzothiazole/benzoxazole derivatives: Design, synthesis, p38α MAP kinase inhibition, anti-inflammatory activity and molecular docking studies.
Tariq, Sana, Kamboj, Payal, Alam, Ozair, Amir, Mohd,
Vol. 81 pp. 630-641
|
2018 |
439
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| 66 |
Synthesis and biological evaluation of myricetin-pentadienone hybrids as potential anti-inflammatory agents in vitro and in vivo.
Liu, Chao, Han, Xu, Yu, Pei Jing, Chen, Liu Zeng, Xue, Wei, Liu, Xin Hua,
Vol. 96 pp. 103597
|
2020 |
392
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| 130 |
Design and synthesis of novel isatin-based derivatives targeting cell cycle checkpoint pathways as potential anticancer agents.
Yousef, Mohamed A, Ali, Ahmed M, El-Sayed, Wael M, Qayed, Wesam S, Farag, Hassan H A, Aboul-Fadl, Tarek,
Vol. 105 pp. 104366
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2020 |
383
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| 6 |
Novel Pyrazoloquinolin-2-ones: Design, synthesis, docking studies, and biological evaluation as antiproliferative EGFR-TK inhibitors.
Elbastawesy, Mohammed A I, Aly, Ashraf A, Ramadan, Mohamed, Elshaier, Yaseen A M M, Youssif, Bahaa G M, Brown, Alan B, El-Din A Abuo-Rahma, Gamal,
Vol. 90 pp. 103045
|
2019 |
375
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| 60 |
Anticancer effects of sodium and potassium quercetin-5'-sulfonates through inhibition of proliferation, induction of apoptosis, and cell cycle arrest in the HT-29 human adenocarcinoma cell line.
Czerwonka, Arkadiusz, Maciołek, Urszula, Kałafut, Joanna, Mendyk, Ewaryst, Kuźniar, Anna, Rzeski, Wojciech,
Vol. 94 pp. 103426
|
2020 |
366
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| 77 |
Synthesis and comparative carbonic anhydrase inhibition of new Schiff's bases incorporating benzenesulfonamide, methanesulfonamide, and methylsulfonylbenzene scaffolds.
El-Azab, Adel S, Abdel-Aziz, Alaa A-M, Bua, Silvia, Nocentini, Alessio, Alanazi, Mohammed M, AlSaif, Nawaf A, Al-Suwaidan, Ibrahim A, Hefnawy, Mohamed M, Supuran, Claudiu T,
Vol. 92 pp. 103225
|
2019 |
365
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| 62 |
Green synthesis of selenium-N-heterocyclic carbene compounds: Evaluation of antimicrobial and anticancer potential.
Kamal, Amna, Nazari V, Mansoureh, Yaseen, Muhammad, Iqbal, Muhammad Adnan, Ahamed, Mohamed B Khadeer, Majid, Aman Shah Abdul, Bhatti, Haq Nawaz,
Vol. 90 pp. 103042
|
2019 |
359
|
| 9 |
Targeting malaria and leishmaniasis: Synthesis and pharmacological evaluation of novel pyrazole-1,3,4-oxadiazole hybrids. Part II
Verma, G.
Vol. 89 pp. 0-0
|
2019 |
352
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| 10 |
Targeting hepatocellular carcinoma: Synthesis of new pyrazole-based derivatives, biological evaluation, DNA binding, and molecular modeling studies
Omran, D.
Vol. 88 pp. 0-0
|
2019 |
346
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