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Keyword Connections
pyrazolopyrimidine
Journals
4
1
Molecules (Basel, Switzerland)
2
Journal of medicinal chemistry
3
chemistry central journal
4
medicinal chemistry (shariqah (united arab emirates))
Research Groups
0
No Research Group Connected
Bibliographies
33
1
The Development of Novel Compounds Against Malaria: Quinolines, Triazolpyridines, Pyrazolopyridines and Pyrazolopyrimidines.
2
Synthesis and Antimicrobial Evaluation of Novel Pyrazolopyrimidines Incorporated with Mono- and Diphenylsulfonyl Groups.
3
Pyrrolopyrazoles: Synthesis, Evaluation and Pharmacological Screening as Antidepressant Agents.
4
Synthesis and anticancer evaluation of some novel pyrimido[5,4-e][1,2,4]triazines and pyrazolo[3,4-d]pyrimidine using DMF-DMA as methylating and cyclizing agent.
5
Development of Potent Inhibitors of Receptor Tyrosine Kinases by Ligand-Based Drug Design and Target-Biased Phenotypic Screening.
6
Design and evaluation of pyrazolopyrimidines as KCNQ channel modulators.
7
Characterization of Covalent Pyrazolopyrimidine-MKK7 Complexes and a Report on a Unique DFG-in/Leu-in Conformation of Mitogen-Activated Protein Kinase Kinase 7 (MKK7).
8
A pyrazolopyrimidine based fluorescent probe for the detection of Cu and Ni and its application in living cells.
9
Design, Synthesis and Antitumor Evaluation of Novel Pyrazolopyrimidines and Pyrazoloquinazolines.
10
Structure-Guided Development of Covalent and Mutant-Selective Pyrazolopyrimidines to Target T790M Drug Resistance in Epidermal Growth Factor Receptor.
11
Novel pyrazolopyrimidines: Synthesis, in vitro cytotoxic activity and mechanistic investigation.
12
The application of bioactive pyrazolopyrimidine unit for the construction of fluorescent biomarkers
13
The development of novel compounds against malaria: Quinolines, triazolpyridines, pyrazolopyridines and pyrazolopyrimidines
14
A Novel Pyrazolopyrimidine Ligand of Human PGK1 and Stress Sensor DJ1 Modulates the Shelterin Complex and Telomere Length Regulation
15
Discovery of pyrazolopyrimidine derivatives as potent BTK inhibitors with effective anticancer activity in MCL
16
New pyrazolopyrimidine derivatives as Leishmania amazonensis arginase inhibitors
17
Development of Potent and Selective Pyrazolopyrimidine IRAK4 Inhibitors
18
COX-1/COX-2 inhibition assays and histopathological study of the new designed anti-inflammatory agent with a pyrazolopyrimidine core
19
Scalable Process Design for a PDE10A Inhibitor Consisting of Pyrazolopyrimidine and Quinoxaline as Key Units
20
Synthesis and characterization of new pyrido- and pyrazolopyrimidine derivatives using 2-substituted vinamidinium salts
21
Dual-response detection of Ni<sup>2+</sup> and Cu<sup>2+</sup> ions by a pyrazolopyrimidine-based fluorescent sensor and the application of this sensor in bioimaging
22
Evaluation of pyrazolopyrimidine derivatives as microtubule affinity regulating kinase 4 inhibitors: Towards therapeutic management of Alzheimer’s disease
23
Synthesis of Some Substituted Pyrazolopyrimidine Derivatives: An Environmentally Benign Approach
24
Pharmacokinetics and in Vivo Efficacy of Pyrazolopyrimidine, Pyrrolopyrimidine, and 5-Aminopyrazole-4-Carboxamide Bumped Kinase Inhibitors against Toxoplasmosis
25
Novel potential pyrazolopyrimidine based translocator protein ligands for the evaluation of neuroinflammation with PET
26
Structural basis of pyrazolopyrimidine derivatives as CAMKIIδ kinase inhibitors: insights from 3D QSAR, docking studies and in silico ADMET evaluation
27
Synthesis and anti-Plasmodium falciparum evaluation of novel pyrazolopyrimidine derivatives
28
Discovery of novel pyrrolopyrimidine/pyrazolopyrimidine derivatives bearing 1,2,3-triazole moiety as c-Met kinase inhibitors
29
Efficient acid catalytic synthesis of pyrazolopyrimidines from 1H-pyrazol-5-yl-N,N-dimethylformamidines with cyanamide
30
Design, synthesis and biological evaluation of novel 3-substituted pyrazolopyrimidine derivatives as potent Bruton's tyrosine kinase (BTK) inhibitors
31
Brønsted Acidic Ionic Liquid-Catalyzed Regioselective Synthesis of Pyrazolopyrimidines and Their Photophysical Properties
32
Trisubstituted pyrazolopyrimidines as novel angiogenesis inhibitors.
33
Synthesis and Isomerization of Some Novel Pyrazolopyrimidine and Pyrazolotriazolopyrimidine Derivatives